SCHEMBL28145809

SCHEMBL28145809

Clc1ccc(CN2CCN(c3ncn[nH]3)CC2)cc1Cl

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.56
POLB P06746 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
LMNA P02545 1/20 0.48
HTR1A P08908 2/20 0.46
HTR2C P28335 2/20 0.46
FAAH O00519 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CACNA1G O43497 3/20 0.42
KCNH2 Q12809 2/20 0.42
OPRL1 P41146 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
TMEM97 Q5BJF2 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
ROCK2 O75116 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28844153 0.85 SIGMAR1 (0.40) SIGMAR1POLBSMN1; SMN2LMNAHTR1A
SCHEMBL28145812 0.82 KDM4E (0.58) HTR1AHTR2CMEN1KMT2AMAPT
SCHEMBL28145820 0.82 LMNA (0.51) LMNAMEN1KMT2AMAPTHTT
SCHEMBL28145836 0.82 PRMT6 (0.47) LMNAMEN1KMT2AMAPTHTT
SCHEMBL28144823 0.78 OPRK1 (0.43) LMNAMEN1KMT2AKCNH2MAPT
SCHEMBL28145787 0.78 ALDH1A1 (0.54) LMNAMEN1KMT2AMAPTHTT
SCHEMBL28144828 0.78 KDM4E (0.56) POLBMEN1KMT2ACYP1A2HTT
SCHEMBL28144854 0.77 HRH3 (0.47) MEN1KMT2AROCK2
SCHEMBL28144851 0.77 PRMT6 (0.56) SIGMAR1LMNAMEN1KMT2AMAPT
SCHEMBL10860653 0.76 SIGMAR1 (0.54) SIGMAR1POLBSMN1; SMN2LMNAHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106659715-A substituted aminotriazoles and methods of use thereof 药物发现研究所 2017-05-10 CN claimed
CN-106659715-A substituted aminotriazoles and methods of use thereof 药物发现研究所 2017-05-10 CN disclosed