SCHEMBL28844153

SCHEMBL28844153

CN(C)c1ccc(CN2CCN(c3ncn[nH]3)CC2)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.40
POLB P06746 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
LMNA P02545 1/20 0.37
TSHR P16473 2/20 0.37
HTT P42858 1/20 0.37
ACHE P22303 1/20 0.36
BACE1 P56817 1/20 0.36
ALDH1A1 P00352 1/20 0.35
DCTPP1 Q9H773 1/20 0.35
HTR1A P08908 1/20 0.35
HTR2C P28335 1/20 0.35
CXCR3 P49682 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28145817 0.86 FAAH (0.37) POLBSMN1; SMN2MEN1KMT2ATSHR
SCHEMBL28145809 0.85 SIGMAR1 (0.56) SIGMAR1POLBSMN1; SMN2MEN1KMT2A
SCHEMBL28145787 0.83 ALDH1A1 (0.54) MEN1KMT2ALMNATSHRHTT
SCHEMBL16826185 0.80 GAA (0.39) SIGMAR1POLBSMN1; SMN2MEN1KMT2A
SCHEMBL28145793 0.77 GALR3 (0.40) SIGMAR1POLBHTTALDH1A1HTR1A
SCHEMBL28145812 0.76 KDM4E (0.58) MEN1KMT2AACHEBACE1HTR1A
SCHEMBL28145836 0.76 PRMT6 (0.47) MEN1KMT2ALMNATSHRHTT
SCHEMBL28145820 0.76 LMNA (0.51) MEN1KMT2ALMNATSHRHTT
SCHEMBL28144823 0.75 OPRK1 (0.43) MEN1KMT2ALMNAALDH1A1DCTPP1
SCHEMBL28144854 0.74 HRH3 (0.47) MEN1KMT2ATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106659715-A substituted aminotriazoles and methods of use thereof 药物发现研究所 2017-05-10 CN claimed
CN-106659715-A substituted aminotriazoles and methods of use thereof 药物发现研究所 2017-05-10 CN disclosed