SCHEMBL28146404

SCHEMBL28146404

C[C](C)CN1CCCC1c1ccc(Br)cc1

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
MAPK1 P28482 1/20 0.42
CYP2C19 P33261 1/20 0.42
OPRM1 P35372 1/20 0.41
OPRK1 P41145 1/20 0.41
CHRNA7 P36544 4/20 0.41
CHRNB2 P17787 2/20 0.41
CHRNA4 P43681 2/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CYP19A1 P11511 2/20 0.39
TSHR P16473 1/20 0.37
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28844433 0.79 ALDH1A1 (0.48)
SCHEMBL29489966 0.79 ATM (0.43) CYP2D6CYP2C9MAPK1CYP2C19CHRNA7
SCHEMBL20680930 0.78 CHRNB2 (0.67) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL1117990 0.78 CHRNB2 (0.67) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL28849366 0.77 TRPV1 (0.45)
SCHEMBL16881226 0.76 CYP2C9 (0.41) CYP2D6CYP2C9MAPK1CYP2C19OPRM1
SCHEMBL3572634 0.76 DRD2 (0.41) CYP2D6CYP2C9MAPK1CYP2C19CHRNA7
SCHEMBL2047049 0.75 HTR1A (0.49) CYP2D6MAPK1CYP2C19OPRM1OPRK1
SCHEMBL1423483 0.74 RIPK1 (0.50) CYP2D6CYP2C9MAPK1CYP2C19ACHE
SCHEMBL29515757 0.74 RIPK1 (0.50) CYP2D6CYP2C9MAPK1CYP2C19ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106661034-A Pyrrolopyrimidines as TLR7 agonists 正大天晴药业集团股份有限公司 2017-05-10 CN disclosed