SCHEMBL28187482

SCHEMBL28187482

COc1ccccc1-c1c(Br)c2ccccc2n1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 5/20 0.48
KDM4E B2RXH2 4/20 0.44
ALDH1A1 P00352 3/20 0.43
GPR3 P46089 1/20 0.41
L3MBTL1 Q9Y468 3/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
HTT P42858 2/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ADORA2A P29274 1/20 0.39
APP P05067 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
LMNA P02545 2/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28191212 0.80 GPR3 (0.47) NTRK1KDM4EALDH1A1GPR3HTT
SCHEMBL9177751 0.77 EGFR (0.51) NTRK1KDM4EALDH1A1L3MBTL1KMT2A
SCHEMBL28186733 0.73 ALDH1A1 (0.57) ALDH1A1GPR3L3MBTL1KMT2AMEN1
SCHEMBL28853473 0.72 NTRK1 (0.39) NTRK1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL14047742 0.70 L3MBTL1 (0.57) NTRK1KDM4EALDH1A1GPR3L3MBTL1
SCHEMBL30648519 0.70 CYP11B2 (0.47) KDM4EALDH1A1KMT2AMEN1HTT
SCHEMBL13890161 0.69 KDM4E (0.58) KDM4EALDH1A1KMT2AMEN1HPGD
SCHEMBL8476766 0.69 KDM4E (0.44) NTRK1KDM4EALDH1A1KMT2AMEN1
SCHEMBL28362345 0.68 APP (0.48) KDM4EALDH1A1L3MBTL1KMT2AMEN1
SCHEMBL5026697 0.68 ALKBH5 (0.59) KDM4EALDH1A1GPR3L3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107445991-A A kind of Phosphine ligands of indoles skeleton and its preparation method and application 香港理工大学深圳研究院 2017-12-08 CN disclosed