SCHEMBL28201586

SCHEMBL28201586

CNCC1=Nc2ncccc2CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.36
ADRB2 P07550 2/20 0.31
HDAC1 Q13547 2/20 0.31
HDAC6 Q9UBN7 2/20 0.31
HRH3 Q9Y5N1 1/20 0.31
CHRM2 P08172 3/20 0.30
CHRM1 P11229 3/20 0.30
DRD2 P14416 3/20 0.30
HTR2A P28223 3/20 0.30
HTR2C P28335 3/20 0.30
ADRA1A P35348 3/20 0.30
HRH1 P35367 3/20 0.30
OPRK1 P41145 3/20 0.30
HTR2B P41595 3/20 0.30
KCNH2 Q12809 3/20 0.30
CYP1A2 P05177 2/20 0.30
CYP3A4 P08684 2/20 0.30
CYP2D6 P10635 2/20 0.30
ADRA2B P18089 2/20 0.30
ADRA2C P18825 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28201595 0.78 L3MBTL1 (0.36) HDAC1HDAC6ADRA2BADRA2CHTT
SCHEMBL28201579 0.77 HRH1 (0.35) ADRB2HRH3CHRM2CHRM1DRD2
SCHEMBL19142282 0.72 CYP11B1 (0.36) CYP2A6CHRM2CHRM1DRD2HTR2A
SCHEMBL28857380 0.70 HRH1 (0.34) ADRB2HDAC1HDAC6CHRM2CHRM1
SCHEMBL4340785 0.70 TSHR (0.32) HDAC1HDAC6CHRM2CHRM1DRD2
SCHEMBL28202178 0.68 HDAC8 (0.32) CHRM2CHRM1DRD2HTR2AHTR2C
SCHEMBL28276888 0.68 CYP11B2 (0.33) CHRM2CHRM1DRD2HTR2AHTR2C
SCHEMBL28195678 0.68 HDAC1 (0.32) HDAC1HDAC6CHRM2CHRM1DRD2
SCHEMBL28201612 0.68 NPC1 (0.33) CHRM2CHRM1DRD2HTR2AHTR2C
SCHEMBL28201589 0.65 CHRM2 (0.30) CHRM2CHRM1DRD2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105683188-B The ring pyridinyl derivatives of condensed ring two as FGFR4 inhibitor 诺华股份有限公司 2018-02-09 CN disclosed