SCHEMBL2825632

SCHEMBL2825632

Cc1nc2c(Br)cccc2c(-c2ccc(F)cc2)c1C(=O)C1CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.37
HTT P42858 3/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
AR P10275 1/20 0.35
NPSR1 Q6W5P4 2/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
PRNP P04156 1/20 0.35
PPARG P37231 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
NR2E3 Q9Y5X4 1/20 0.35
NCOR2 Q9Y618 1/20 0.35
ALDH1A1 P00352 3/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C19 P33261 2/20 0.34
HPGD P15428 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2825469 0.90 GAA (0.45) KDM4EMEN1KMT2ANPSR1GAA
SCHEMBL2829123 0.82 ENPP1 (0.40) HTTKDM4EMEN1KMT2ANPSR1
SCHEMBL2821075 0.78 PRNP (0.59) HTTPRNPPPARGRXFP1NR2E3
SCHEMBL2823585 0.73 ALDH1A1 (0.61) HTTKDM4EMEN1KMT2ANPSR1
SCHEMBL2821517 0.72 NPSR1 (0.67) HTTKDM4EMEN1KMT2ANPSR1
SCHEMBL2821493 0.72 MAPT (0.46) KDM4EMEN1KMT2ANPSR1GAA
SCHEMBL2821849 0.72 GAA (0.46) ESR1KDM4EMEN1KMT2ANPSR1
SCHEMBL2823193 0.71 FABP3 (0.45) HTTKDM4EMEN1KMT2ANPSR1
SCHEMBL2825660 0.70 NR1H2 (0.41)
SCHEMBL2824583 0.70 NCF1 (0.43) HTTKDM4EMEN1KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809605-B1 QUINOLINES AS ALLOSTERIC ENHANCERS OF THE GABA-B RECEPTORS HOFFMANN LA ROCHE (CH) 2010-08-11 EP claimed