SCHEMBL28264167

SCHEMBL28264167

CC(=O)C(c1ccc(N(C)C)cc1)c1c(F)cccc1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
MAT2A P31153 1/20 0.41
KCNH2 Q12809 1/20 0.41
KMT2A Q03164 2/20 0.40
GAA P10253 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KDM4E B2RXH2 2/20 0.39
MAPT P10636 4/20 0.38
HPGD P15428 2/20 0.38
RAB9A P51151 3/20 0.38
NPC1 O15118 2/20 0.38
CNR2 P34972 1/20 0.38
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
MEN1 O00255 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
JAK3 P52333 1/20 0.36
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14741002 0.78 ALDH1A1 (0.56) ALDH1A1KMT2AGAAL3MBTL1KDM4E
SCHEMBL7541462 0.76 KCNH2 (0.47) ALDH1A1MAT2AKCNH2KMT2AGAA
SCHEMBL28118171 0.72 THRB (0.35) ALDH1A1GAAKDM4EMAPTHPGD
SCHEMBL13170115 0.70 CES2 (0.62) KMT2AHPGDCES2CES1MEN1
SCHEMBL8812406 0.70 ALDH1A1 (0.59) ALDH1A1KMT2AGAAL3MBTL1KDM4E
SCHEMBL27872658 0.70 RAB9A (0.49) ALDH1A1KMT2AGAAKDM4EMAPT
SCHEMBL10818690 0.68 ALDH1A1 (0.59) ALDH1A1KMT2AGAAL3MBTL1KDM4E
SCHEMBL11304149 0.67 ALDH1A1 (0.56) ALDH1A1KMT2AGAAL3MBTL1KDM4E
SCHEMBL5983400 0.67 ALDH1A1 (0.46) ALDH1A1KCNH2KMT2AL3MBTL1KDM4E
SCHEMBL11330475 0.66 L3MBTL1 (0.43) ALDH1A1KMT2AL3MBTL1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109096178-A Phenylethynyl substituted benzenes and heterocycles useful for the treatment of cancer and uses thereof 肯塔基大学研究基金会 2018-12-28 CN disclosed