SCHEMBL2826464

SCHEMBL2826464

Cc1cccc(NC(=O)Oc2ncsc2Nc2cccc(C#N)c2)n1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.58
RAB9A P51151 5/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
GRM5 P41594 3/20 0.51
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
SYK P43405 1/20 0.41
ABCG2 Q9UNQ0 2/20 0.40
SLC2A1 P11166 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
GBA1 P04062 2/20 0.39
CDK4 P11802 1/20 0.39
CDK2 P24941 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2829479 0.89 NPC1 (0.43) NPC1RAB9ASMN1; SMN2GRM5ALDH1A1
SCHEMBL2829743 0.88 NPC1 (0.42) NPC1RAB9ASMN1; SMN2GRM5ABCG2
SCHEMBL2830126 0.86 NPC1 (0.42) NPC1RAB9ASMN1; SMN2GRM5LMNA
SCHEMBL2830797 0.86 RAB9A (0.51) NPC1RAB9ASMN1; SMN2GRM5MEN1
SCHEMBL2826737 0.85 RAB9A (0.56) NPC1RAB9ASMN1; SMN2GRM5MEN1
SCHEMBL2824780 0.85 ALDH1A1 (0.44) NPC1RAB9ASMN1; SMN2ALDH1A1MEN1
SCHEMBL2826324 0.84 NPC1 (0.58) NPC1RAB9ASMN1; SMN2GRM5ALDH1A1
SCHEMBL2830129 0.84 CYP1A2 (0.44) NPC1RAB9ASMN1; SMN2GRM5ALDH1A1
SCHEMBL2825977 0.82 GRM5 (0.50) NPC1RAB9ASMN1; SMN2GRM5MEN1
SCHEMBL2828556 0.81 MAOB (0.46) NPC1RAB9AALDH1A1LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844044-B1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-07-21 EP claimed