SCHEMBL2830126

SCHEMBL2830126

Cc1csc(NC(=O)Oc2ncsc2Nc2cccc(C#N)c2)n1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.42
RAB9A P51151 4/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
HPGD P15428 2/20 0.41
GCK P35557 5/20 0.40
POLB P06746 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GRM4 Q14833 1/20 0.40
SMARCA2 P51531 1/20 0.39
SMARCA4 P51532 1/20 0.39
GRM5 P41594 1/20 0.39
ALOX15 P16050 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2826464 0.86 NPC1 (0.58) NPC1RAB9ASMN1; SMN2MEN1LMNA
SCHEMBL2829743 0.85 NPC1 (0.42) NPC1RAB9ASMN1; SMN2MEN1MAPT
SCHEMBL2828877 0.85 RAB9A (0.52) NPC1RAB9ASMN1; SMN2MEN1LMNA
SCHEMBL2824780 0.84 ALDH1A1 (0.44) NPC1RAB9ASMN1; SMN2MEN1MAPT
SCHEMBL2828556 0.81 MAOB (0.46) NPC1RAB9AMEN1LMNAMAPT
SCHEMBL2824997 0.81 GRM5 (0.48) NPC1RAB9ASMN1; SMN2MAPTHPGD
SCHEMBL2829479 0.80 NPC1 (0.43) NPC1RAB9ASMN1; SMN2MEN1MAPT
SCHEMBL2829552 0.78 RAB9A (0.47) NPC1RAB9ASMN1; SMN2MEN1LMNA
SCHEMBL2827802 0.77 SCD (0.48) NPC1RAB9ASMN1; SMN2MEN1MAPT
SCHEMBL2826277 0.75 NPC1 (0.40) NPC1RAB9ASMN1; SMN2MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844044-B1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-07-21 EP claimed