SCHEMBL28274202

SCHEMBL28274202

O=CNc1nc(Cl)c2ccccc2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
METAP1 P53582 1/20 0.41
ALDH1A1 P00352 4/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
NPY5R Q15761 3/20 0.39
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
KDM4E B2RXH2 4/20 0.38
MAPT P10636 3/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
TAAR1 Q96RJ0 2/20 0.38
HPGD P15428 1/20 0.38
ALOX12 P18054 1/20 0.38
TDP1 Q9NUW8 2/20 0.38
TLR8 Q9NR97 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27962998 0.79 ALDH1A1 (0.50) ALDH1A1MEN1KMT2AMAPTNPC1
SCHEMBL5505630 0.78 TYMS (0.39) KMT2AMAPTGAA
SCHEMBL12496376 0.77 ALDH1A1 (0.41) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL3337224 0.77 NUDT1 (0.61) MAOAMAOBMETAP1PDE4APDE4B
SCHEMBL1980544 0.75 IGF1R (0.52) MAOAMAOBALDH1A1MEN1KMT2A
SCHEMBL12495765 0.73 ADH1B (0.38) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL28212751 0.73 ADORA3 (0.61) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL27845963 0.73 MAOA (0.47) MAOAMAOBMETAP1ALDH1A1PDE4A
SCHEMBL24287271 0.72 KDM4E (0.59) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL29516515 0.72 KDM4E (0.59) ALDH1A1MEN1KMT2AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106008373-B Disubstituted bicyclic derivative and its application as efflux pump inhibitor in antibacterial 山东大学 2019-02-22 CN disclosed