SCHEMBL2828532

SCHEMBL2828532

CCNc1scnc1OC(=O)Nc1nc(C)cs1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
MAPT P10636 2/20 0.44
ALDH1A1 P00352 1/20 0.44
RAB9A P51151 7/20 0.42
HPGD P15428 1/20 0.42
GCK P35557 1/20 0.42
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
POLB P06746 2/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 1/20 0.41
GRM5 P41594 1/20 0.41
SMARCA2 P51531 1/20 0.40
SMARCA4 P51532 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2826011 0.84 ALDH1A1 (0.41) NPC1KMT2ASMN1; SMN2MAPTALDH1A1
SCHEMBL2828968 0.83 MAPT (0.44) NPC1SMN1; SMN2MAPTALDH1A1RAB9A
SCHEMBL2828877 0.80 RAB9A (0.52) NPC1KMT2ASMN1; SMN2MAPTALDH1A1
SCHEMBL2827802 0.78 SCD (0.48) NPC1KMT2ASMN1; SMN2MAPTALDH1A1
SCHEMBL2829552 0.78 RAB9A (0.47) NPC1KMT2ASMN1; SMN2MAPTRAB9A
SCHEMBL2830217 0.77 RAB9A (0.41) NPC1SMN1; SMN2MAPTALDH1A1RAB9A
SCHEMBL2824997 0.76 GRM5 (0.48) NPC1SMN1; SMN2MAPTRAB9AHPGD
SCHEMBL11183549 0.74 MAPT (0.57) NPC1KMT2ASMN1; SMN2MAPTALDH1A1
SCHEMBL2830832 0.74 ALDH1A1 (0.49) NPC1KMT2ASMN1; SMN2MAPTALDH1A1
SCHEMBL2827794 0.73 CHRNB2 (0.45) NPC1SMN1; SMN2MAPTRAB9ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844044-B1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-07-21 EP claimed