SCHEMBL2829067

SCHEMBL2829067

CCn1nccc1Nc1sc(C)nc1OC(=O)Nc1ccnc(C)n1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSK P43235 2/20 0.35
SORT1 Q99523 4/20 0.34
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
PIK3C3 Q8NEB9 3/20 0.32
GRM5 P41594 1/20 0.31
PIK3CA P42336 1/20 0.31
RIPK1 Q13546 1/20 0.31
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
NTRK1 P04629 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2832743 0.87 SORT1 (0.34) CTSKSORT1ALDH1A1KMT2APIK3C3
SCHEMBL5185611 0.83 GRM5 (0.43) SORT1ALDH1A1MEN1KMT2APIK3C3
SCHEMBL2826529 0.80 SMN1; SMN2 (0.36) SORT1MEN1KMT2APIK3C3GRM5
SCHEMBL2830005 0.79 SORT1 (0.35) CTSKSORT1ALDH1A1KMT2AGRM5
SCHEMBL2829035 0.78 AURKB (0.37) GRM5
SCHEMBL2826030 0.78 PIK3CA (0.37) SORT1ALDH1A1PIK3CARIPK1NPC1
SCHEMBL2830257 0.77 GRM5 (0.50) SORT1KMT2APIK3C3GRM5NTRK1
SCHEMBL2826649 0.77 HTR2C (0.36) SORT1ALDH1A1PIK3C3GRM5RIPK1
SCHEMBL2833176 0.77 SORT1 (0.41) SORT1PIK3C3GRM5PIK3CANPC1
SCHEMBL2829325 0.77 JAK2 (0.41) SORT1MEN1KMT2APIK3C3NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844044-B1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-07-21 EP claimed