SCHEMBL28294262

SCHEMBL28294262

N#Cc1ccc(CN2Cc3ccccc3CC2C(N)=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.44
MMP8 P22894 2/20 0.43
MMP3 P08254 1/20 0.43
NAMPT P43490 1/20 0.42
HSD11B1 P28845 1/20 0.42
HTR1A P08908 3/20 0.42
HTR7 P34969 3/20 0.42
MAPT P10636 2/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PRMT5 O14744 7/20 0.41
WDR77 Q9BQA1 7/20 0.41
FNTA P49354 1/20 0.40
FNTB P49356 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6920539 0.81 HTR1A (0.50) OPRM1MMP3HTR1AHTR7
SCHEMBL29870443 0.74 ACE (0.49) MMP8MMP3LMNAPOLBL3MBTL1
SCHEMBL8336724 0.74 ACE (0.49) MMP8MMP3LMNAPOLBL3MBTL1
SCHEMBL7478005 0.74 ACE (0.49) MMP8MMP3LMNAPOLBL3MBTL1
SCHEMBL5900780 0.74 HSD11B1 (0.61) MMP8HSD11B1POLB
SCHEMBL18953046 0.73 SIRT2 (0.45) MMP8MMP3HTR1AHTR7KDM4E
Hydrochloric Acid SCHEMBL5901272 0.73 HSD11B1 (0.60) MMP8HSD11B1POLB
SCHEMBL8342126 0.73 MMP8 (0.58) MMP8MMP3POLBL3MBTL1
SCHEMBL8342131 0.73 MMP8 (0.58) MMP8MMP3POLBL3MBTL1
SCHEMBL7477932 0.73 FNTA (0.56) FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109776414-A A kind of Bcl-2 protein inhibitor and its preparation method and application 山东大学 2019-05-21 CN disclosed