SCHEMBL6920539

SCHEMBL6920539

COc1ccc(CN2Cc3ccccc3CC2C(N)=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.50
HTR7 P34969 2/20 0.50
HDAC8 Q9BY41 1/20 0.50
SIRT2 Q8IXJ6 1/20 0.48
SIRT1 Q96EB6 1/20 0.48
DRD2 P14416 3/20 0.47
DRD4 P21917 3/20 0.47
ALDH1A1 P00352 1/20 0.46
MMP9 P14780 7/20 0.45
MMP1 P03956 4/20 0.45
MMP3 P08254 3/20 0.45
ADAM17 P78536 3/20 0.45
ADAM9 Q13443 2/20 0.45
AREG P15514 1/20 0.44
TNF P01375 1/20 0.44
NOD2 Q9HC29 1/20 0.44
NOD1 Q9Y239 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
OPRM1 P35372 1/20 0.44
MAOB P27338 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6920302 0.89 HDAC8 (0.53) HDAC8MMP9MMP1MMP3ADAM17
SCHEMBL6820388 0.85 HDAC8 (0.48) HDAC8MMP9MMP1MMP3ADAM17
SCHEMBL28294262 0.81 OPRM1 (0.44) HTR1AHTR7MMP3OPRM1
SCHEMBL7127952 0.79 SIGMAR1 (0.47) SIGMAR1OPRM1
SCHEMBL32677056 0.77 HTR1A (0.44) HTR1AHTR7MMP9OPRM1
SCHEMBL7533950 0.76 KDM4E (0.50) HTR1AHDAC8SIRT2SIRT1DRD4
SCHEMBL7533954 0.76 KDM4E (0.50) HTR1AHDAC8SIRT2SIRT1DRD4
SCHEMBL8383113 0.75 GP6 (0.63) ALDH1A1MMP3
SCHEMBL7478005 0.74 ACE (0.49) ALDH1A1MMP3
SCHEMBL29870443 0.74 ACE (0.49) ALDH1A1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004041816-A1 AZACYCLIC COMPOUNDS AS OREXIN RECEPTOR ANTAGONIST GLAXO GROUP LIMITED (GB) 2004-05-21 WO disclosed