SCHEMBL28294415

SCHEMBL28294415

COc1cnc2c(Cl)cccc2c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC40A1 Q9NP59 2/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
PIK3CD O00329 4/20 0.42
RELA Q04206 1/20 0.42
HPGDS O60760 2/20 0.42
PARP1 P09874 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2A6 P11509 1/20 0.41
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
NFE2L2 Q16236 2/20 0.39
BACE2 Q9Y5Z0 1/20 0.38
NQO2 P16083 1/20 0.38
PIN1 Q13526 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Jineol Methyl Ether SCHEMBL8613544 0.81 HPGDS (0.62) MEN1KMT2ARELAHPGDSPARP1
SCHEMBL29923835 0.81 MAPT (0.45) SLC40A1KMT2APIK3CDRELAHPGDS
SCHEMBL4799696 0.80 NR1H2 (0.44) MEN1KMT2ACYP1A2NPC1RAB9A
SCHEMBL10320559 0.79 PARP1 (0.45) SLC40A1MEN1KMT2ARELAHPGDS
SCHEMBL15703131 0.79 PSMD14 (0.62) RELAHPGDSPARP1CYP1A2CYP2A6
SCHEMBL6347577 0.79 RELA (0.52) RELACYP1A2CYP2A6NPC1RAB9A
SCHEMBL30492638 0.79 RELA (0.52) RELACYP1A2CYP2A6NPC1RAB9A
SCHEMBL6422325 0.77 PSMD14 (0.62) SLC40A1PARP1CYP1A2CYP2A6
SCHEMBL1408873 0.76 CYP1A2 (0.50) MEN1KMT2ARELACYP1A2CYP2A6
SCHEMBL6356302 0.76 CCR1 (0.62) SLC40A1MEN1KMT2ARELACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed