SCHEMBL29923835

SCHEMBL29923835

COc1cnc2c(C)cccc2c1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.45
KDM4E B2RXH2 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
PIK3CD O00329 5/20 0.43
HPGDS O60760 1/20 0.43
RELA Q04206 1/20 0.43
PARP1 P09874 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP2A6 P11509 2/20 0.42
PSMD14 O00487 1/20 0.42
COPS5 Q92905 1/20 0.42
MGAM O43451 2/20 0.40
GAA P10253 2/20 0.40
SI P14410 2/20 0.40
MGAM2 Q2M2H8 2/20 0.40
KMT2A Q03164 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SLC40A1 Q9NP59 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Jineol Methyl Ether SCHEMBL8613544 0.82 HPGDS (0.62) MAPTKDM4EHPGDSRELAPARP1
SCHEMBL28294415 0.81 SLC40A1 (0.44) PIK3CDHPGDSRELAPARP1CYP1A2
SCHEMBL15703131 0.81 PSMD14 (0.62) KDM4EHPGDSRELAPARP1CYP1A2
SCHEMBL10320559 0.81 PARP1 (0.45) MAPTKDM4EHPGDSRELAPARP1
SCHEMBL30492638 0.81 RELA (0.52) RELACYP1A2CYP2A6NPC1RAB9A
SCHEMBL6347577 0.81 RELA (0.52) RELACYP1A2CYP2A6NPC1RAB9A
SCHEMBL1408873 0.77 CYP1A2 (0.50) MAPTL3MBTL1RELACYP1A2CYP2A6
SCHEMBL30492598 0.77 CCR1 (0.62) MAPTKDM4EL3MBTL1RELACYP1A2
SCHEMBL6356302 0.77 CCR1 (0.62) MAPTKDM4EL3MBTL1RELACYP1A2
SCHEMBL7376462 0.77 PSMD14 (0.67) KDM4EPARP1CYP1A2CYP2A6PSMD14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed