SCHEMBL2829476

SCHEMBL2829476

Cc1noc(C)c1Nc1scnc1OC(=O)Nc1cccc(Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.48
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
LMNA P02545 3/20 0.43
HTT P42858 2/20 0.43
NPC1 O15118 6/20 0.42
RAB9A P51151 6/20 0.42
ATM Q13315 1/20 0.42
AURKA O14965 1/20 0.42
AURKB Q96GD4 1/20 0.42
MAPT P10636 6/20 0.41
ALDH1A1 P00352 3/20 0.41
PLA2G1B P04054 1/20 0.41
ATG4B Q9Y4P1 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
POLB P06746 1/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2829439 0.90 ALDH1A1 (0.43) AKR1C3MEN1KMT2ANPC1RAB9A
SCHEMBL2826420 0.84 LMNA (0.47) MEN1KMT2ALMNAHTTNPC1
SCHEMBL2830058 0.83 LMNA (0.50) MEN1KMT2ALMNAHTTNPC1
SCHEMBL2828993 0.82 MAPT (0.51) AKR1C3MEN1KMT2ALMNAHTT
SCHEMBL2827687 0.81 MEN1 (0.49) MEN1KMT2ALMNAHTTNPC1
SCHEMBL2824592 0.80 RAB9A (0.41) MEN1KMT2ALMNANPC1RAB9A
SCHEMBL2829161 0.80 HPGD (0.50) MEN1KMT2ALMNAHTTNPC1
SCHEMBL2826800 0.79 CHRNB2 (0.35) LMNANPC1RAB9AAURKBALDH1A1
SCHEMBL2826660 0.79 LMNA (0.46) MEN1KMT2ALMNAHTTNPC1
SCHEMBL2829084 0.78 HPGD (0.48) MEN1KMT2ALMNAHTTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844044-B1 THIAZOLE-4-CARBOXAMIDE DERIVATIVES AS MGLUR5 ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-07-21 EP claimed