SCHEMBL28297314

SCHEMBL28297314

O=CNN1CCNc2ccccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 3/20 0.38
BRPF1 P55201 1/20 0.37
PIM1 P11309 1/20 0.35
BRD4 O60885 1/20 0.35
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
KMT2A Q03164 1/20 0.34
GPBAR1 Q8TDU6 1/20 0.34
MMP2 P08253 2/20 0.33
MKNK1 Q9BUB5 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
HSD11B1 P28845 1/20 0.32
AVPR2 P30518 1/20 0.32
MMP9 P14780 1/20 0.32
ADAM17 P78536 1/20 0.32
HSD17B3 P37058 1/20 0.32
MAPK1 P28482 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5458675 0.84 BRPF1 (0.40) BRPF1BRD4MEN1GAAKMT2A
SCHEMBL1862935 0.75 AVPR1A (0.46) AVPR1ABRPF1PIM1BRD4GAA
SCHEMBL94614 0.74 SMN1; SMN2 (0.41) AVPR1ABRPF1PIM1BRD4MEN1
SCHEMBL9828967 0.72 AVPR1A (0.40) AVPR1ABRPF1PIM1MEN1GAA
SCHEMBL1383225 0.70 ALDH1A1 (0.44) MEN1GAAKMT2AHPGD
SCHEMBL11070863 0.70
SCHEMBL7757772 0.69 ADRA2A (0.46)
SCHEMBL28833094 0.69 BRD4 (0.41) AVPR1ABRPF1PIM1BRD4MEN1
SCHEMBL3661398 0.68 MAPK1 (0.50) AVPR1APIM1MEN1KMT2AMAPK1
SCHEMBL31512482 0.68 AVPR1A (0.39) AVPR1ABRPF1PIM1BRD4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106029076-B Benzo piperazine composition as BET bromine domain inhibitor 福马疗法公司 2019-06-07 CN disclosed