SCHEMBL28314925

SCHEMBL28314925

CC(C)(C)C(=O)ON1CCC(C)(C(=O)Nc2c(F)cccc2F)CC1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.40
ALDH1A1 P00352 4/20 0.35
CETP P11597 3/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
OPRL1 P41146 1/20 0.35
NLRP3 Q96P20 1/20 0.34
NOX1 Q9Y5S8 1/20 0.34
AVPR2 P30518 3/20 0.33
XIAP P98170 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20137885 0.81 TSHR (0.44) RET
SCHEMBL20069163 0.79 OPRD1 (0.40) RETALDH1A1CETPOPRM1OPRD1
SCHEMBL20158642 0.76 OPRM1 (0.46) RETALDH1A1CETPOPRM1OPRD1
SCHEMBL20205744 0.74 OPRM1 (0.44) RETALDH1A1CETPOPRM1OPRD1
Tert-Butyl Formate SCHEMBL28314926 0.71 RET (0.35) RETALDH1A1CETPNLRP3NOX1
SCHEMBL27796299 0.69 OPRL1 (0.41) OPRM1OPRD1OPRK1OPRL1
SCHEMBL27789518 0.69
SCHEMBL27797082 0.68 CHRM3 (0.40) OPRM1OPRD1OPRK1
SCHEMBL28844207 0.68 RBP4 (0.48) ALDH1A1
SCHEMBL23290589 0.68 GPR119 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110177786-A Pyrazolo [1,5-A] pyridine compounds being substituted are as RET kinase inhibitor 阿雷生物药品公司 2019-08-27 CN disclosed