SCHEMBL28345508

SCHEMBL28345508

O=C1CCSc2sc(C(=O)N3CCN(Cc4ccc(-c5ccc(Cl)cc5)cc4)CC3)cc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LSS P48449 2/20 0.48
GPR183 P32249 1/20 0.44
TP53 P04637 1/20 0.43
PTGS2 P35354 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HRH3 Q9Y5N1 2/20 0.42
TACR3 P29371 1/20 0.42
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 1/20 0.41
AKR1C3 P42330 1/20 0.41
POLB P06746 1/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 2/20 0.40
TSHR P16473 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
CHRM1 P11229 1/20 0.40
HTR2A P28223 1/20 0.40
MCHR1 Q99705 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28397524 0.82 ALDH1A1 (0.46) SMN1; SMN2ALDH1A1AKR1C3POLBLMNA
SCHEMBL28345520 0.82 LSS (0.46) LSSGPR183TP53PTGS2HRH3
SCHEMBL28396249 0.76 MAPT (0.56) TP53SMN1; SMN2ALDH1A1LMNAMAPT
SCHEMBL28348405 0.76 HRH4 (0.47) TP53ALDH1A1KDM4ELMNAMAPT
SCHEMBL28396620 0.75 POLB (0.48) SMN1; SMN2ALDH1A1AKR1C3POLBLMNA
SCHEMBL28400986 0.73 HPGD (0.50) SMN1; SMN2ALDH1A1KDM4EMAPTTSHR
SCHEMBL28393540 0.73 KMT2A (0.55) TP53ALDH1A1POLBLMNAMAPT
SCHEMBL28888486 0.72 L3MBTL1 (0.45) TP53ALDH1A1KDM4EAKR1C3POLB
SCHEMBL28394262 0.72 L3MBTL1 (0.43) TP53ALDH1A1KDM4EAKR1C3POLB
SCHEMBL28394808 0.72 GAA (0.51) SMN1; SMN2ALDH1A1KDM4EPOLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108822125-B 1- (thieno [2,3-b ] thiopyranoformyl) -4-aliphatic alkyl piperazine compound and medical application thereof 沈阳药科大学 2020-01-31 CN claimed
CN-108822125-B 1- (thieno [2,3-b ] thiopyranoformyl) -4-aliphatic alkyl piperazine compound and medical application thereof 沈阳药科大学 2020-01-31 CN disclosed