SCHEMBL28360758

SCHEMBL28360758

O=C(C=Cc1ccc(-c2cc(=O)oc3ccccc23)cc1)C=Cc1ccccn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
HPGD P15428 3/20 0.40
USP2 O75604 1/20 0.40
CA9 Q16790 3/20 0.40
AKR1B1 P15121 2/20 0.40
TUBB4A P04350 2/20 0.40
TUBB P07437 2/20 0.40
TUBA3C P0DPH7 2/20 0.40
TUBA1B P68363 2/20 0.40
TUBA4A P68366 2/20 0.40
TUBB4B P68371 2/20 0.40
TUBB3 Q13509 2/20 0.40
TUBB2A Q13885 2/20 0.40
TUBB8 Q3ZCM7 2/20 0.40
TUBA3E Q6PEY2 2/20 0.40
TUBA1A Q71U36 2/20 0.40
TUBA1C Q9BQE3 2/20 0.40
TUBB6 Q9BUF5 2/20 0.40
TUBB2B Q9BVA1 2/20 0.40
TUBB1 Q9H4B7 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28360755 0.87 CA9 (0.49) ALDH1A1HPGDUSP2CA9AKR1B1
SCHEMBL28756601 0.86 TUBB4A (0.47) ALDH1A1HPGDCA9AKR1B1TUBB4A
SCHEMBL28360775 0.84 HSD11B1 (0.50) ALDH1A1HPGDUSP2CA9AKR1B1
SCHEMBL28356945 0.84 CA9 (0.53) ALDH1A1HPGDUSP2CA9AKR1B1
SCHEMBL28360812 0.84 NPC1 (0.53) USP2CA9AKR1B1CA12ALDH2
SCHEMBL28360763 0.83 TXNRD1 (0.40) ALDH1A1HPGDCA9AKR1B1TUBB4A
SCHEMBL28357051 0.80 ALDH1A1 (0.43) ALDH1A1HPGDUSP2CA9AKR1B1
SCHEMBL28356929 0.80 KMT2A (0.49) ALDH1A1HPGDUSP2CA9AKR1B1
SCHEMBL28356950 0.79 TUBB4A (0.54) ALDH1A1HPGDCA9TUBB4ATUBB
SCHEMBL28360752 0.78 NFE2L2 (0.53) ALDH1A1HPGDTUBB4ATUBBTUBA3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106928176-B Coumarin-containing 1, 4-pentadiene-3-ketone derivative and preparation method and application thereof 贵州大学 2020-02-18 CN disclosed