SCHEMBL28455283

SCHEMBL28455283

CCNc1ccccc1C(=O)N(C)C

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 3/20 0.56
ADRA1A P35348 3/20 0.56
ADRA1B P35368 3/20 0.56
POLB P06746 1/20 0.49
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CXCR2 P25025 7/20 0.47
CXCR1 P25024 3/20 0.44
FABP4 P15090 1/20 0.43
KEAP1 Q14145 1/20 0.42
MASP2 O00187 1/20 0.42
KDM4E B2RXH2 1/20 0.42
GLA P06280 1/20 0.42
MAPT P10636 1/20 0.42
JAK2 O60674 1/20 0.42
JAK1 P23458 1/20 0.42
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28454558 0.86 ADRA1A (0.53) ADRA1DADRA1AADRA1BPOLBMEN1
SCHEMBL28454648 0.84 ADRA1A (0.59) ADRA1DADRA1AADRA1BSMN1; SMN2FABP4
SCHEMBL29212431 0.81 ADRA1D (0.52) ADRA1DADRA1AADRA1BPOLBMEN1
SCHEMBL2001238 0.81 FABP4 (0.48) ADRA1DADRA1AADRA1BPOLBKMT2A
SCHEMBL18657136 0.80 HDAC6 (0.48) ADRA1DADRA1AADRA1BMAPTTP53
SCHEMBL184136 0.79 ALDH1A1 (0.62) POLBMEN1KMT2ASMN1; SMN2FABP4
SCHEMBL6088062 0.79 JAK2 (0.48) ADRA1DADRA1AADRA1BPOLBFABP4
SCHEMBL8343253 0.79 POLB (0.58) ADRA1DADRA1AADRA1BPOLBMEN1
SCHEMBL8828501 0.79 ADRA1D (0.50) ADRA1DADRA1AADRA1BPOLBMEN1
SCHEMBL11520956 0.78 FABP4 (0.49) ADRA1DADRA1AADRA1BPOLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114516855-A Preparation of pyridylpyrazole amide compounds and intermediates therefor 湖南化工研究院有限公司 2022-05-20 CN claimed
CN-114516854-A Preparation method of 1-pyridyl pyrazole amide compound and intermediate thereof 湖南化工研究院有限公司 2022-05-20 CN claimed
CN-111662269-B 1-pyridyl pyrazole amide compound and preparation method and application thereof 湖南化工研究院有限公司 2021-05-07 CN claimed
CN-111662269-A 1-pyridyl pyrazole amide compound and preparation method and application thereof 湖南化工研究院有限公司 2020-09-15 CN claimed
CN-114516855-A Preparation of pyridylpyrazole amide compounds and intermediates therefor 湖南化工研究院有限公司 2022-05-20 CN disclosed
CN-114516854-A Preparation method of 1-pyridyl pyrazole amide compound and intermediate thereof 湖南化工研究院有限公司 2022-05-20 CN disclosed
CN-111662269-B 1-pyridyl pyrazole amide compound and preparation method and application thereof 湖南化工研究院有限公司 2021-05-07 CN disclosed
CN-111662269-A 1-pyridyl pyrazole amide compound and preparation method and application thereof 湖南化工研究院有限公司 2020-09-15 CN disclosed