SCHEMBL28484148

SCHEMBL28484148

Cc1cc2c(C#N)cccc2n1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 1/20 0.43
EGFR P00533 1/20 0.40
SRC P12931 1/20 0.40
TSHR P16473 1/20 0.39
KDM4E B2RXH2 3/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MAOA P21397 3/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
GPR3 P46089 1/20 0.38
ALKBH5 Q6P6C2 1/20 0.37
FTO Q9C0B1 1/20 0.37
VCP P55072 1/20 0.36
NQO2 P16083 1/20 0.36
ALDH1A1 P00352 2/20 0.36
DHFR P00374 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18000161 0.82 HSD17B10 (0.38) EGFRSRCKDM4ECASP1CASP7
SCHEMBL28229252 0.81 IMPDH2 (0.39) IMPDH2TSHRKDM4EHSD17B10VCP
SCHEMBL1429109 0.77 HPGD (0.54) IMPDH2EGFRSRCKDM4EHSD17B10
SCHEMBL13548554 0.75 ALKBH5 (0.52) KDM4ECASP1CASP7HSD17B10CYP1A2
SCHEMBL18028323 0.72 BCHE (0.43) IMPDH2EGFRSRCKDM4EMAOA
SCHEMBL18000262 0.72 GPR3 (0.46) KDM4ECASP1CASP7HSD17B10CYP1A2
SCHEMBL18000203 0.72 GPR3 (0.41) TSHRKDM4ECASP1CASP7HSD17B10
SCHEMBL30622575 0.72 GPR3 (0.46) KDM4ECASP1CASP7HSD17B10CYP1A2
SCHEMBL1355293 0.72 DHFR (0.45) TSHRKDM4ECASP1CASP7HSD17B10
SCHEMBL17680605 0.72 GPR3 (0.41) KDM4ECASP1CASP7HSD17B10CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107820494-B Nuclear receptor modulators 艾伯维公司 2020-10-16 CN disclosed