SCHEMBL28486272

SCHEMBL28486272

CCCCCC(CCCC)(CCCC)CCNCc1ccc(OC(N)=O)nc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 16/20 0.42
S1PR3 Q99500 16/20 0.42
S1PR2 O95136 14/20 0.42
S1PR4 O95977 4/20 0.42
OPRM1 P35372 3/20 0.39
OPRD1 P41143 3/20 0.39
OPRK1 P41145 3/20 0.39
CD274 Q9NZQ7 1/20 0.38
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A3 Q01959 1/20 0.38
GRIN1 Q05586 1/20 0.38
KCNH2 Q12809 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
ROCK1 Q13464 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
LPAR2 Q9HBW0 10/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28486270 0.93 OPRM1 (0.42) S1PR1S1PR3S1PR2S1PR4OPRM1
SCHEMBL28486275 0.81 S1PR1 (0.38) S1PR1S1PR3S1PR2S1PR4OPRM1
SCHEMBL28478495 0.80 OPRM1 (0.40) S1PR1S1PR3S1PR2S1PR4OPRM1
SCHEMBL28482119 0.76 SMN1; SMN2 (0.44) OPRM1OPRD1OPRK1CD274GRIN2D
SCHEMBL11115121 0.74 NFKB1 (0.55)
SCHEMBL28481490 0.70 KMT2A (0.52) OPRM1OPRD1OPRK1CD274GRIN2D
SCHEMBL4687699 0.69 KDM4E (0.54) S1PR1S1PR3S1PR2LPAR2
SCHEMBL3265195 0.68 MEN1 (0.50) S1PR1S1PR3S1PR2LPAR2
SCHEMBL22978445 0.67 GABRP (0.40) OPRM1OPRD1OPRK1CD274GRIN2D
SCHEMBL28375723 0.67 GABRP (0.40) OPRM1OPRD1OPRK1GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111936466-A Compounds for the treatment of cardiac arrhythmias and heart failure 埃利克斯生物技术公司 2020-11-13 CN disclosed