SCHEMBL2850131

SCHEMBL2850131

COc1ccc(-n2ncc(OC(=O)Nc3ccccc3)c2C)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 8/20 0.61
NPC1 O15118 7/20 0.61
PKM P14618 1/20 0.61
ALDH1A1 P00352 4/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
GAA P10253 1/20 0.58
HTT P42858 1/20 0.58
MAPT P10636 5/20 0.56
NFKB1 P19838 1/20 0.56
NFKB2 Q00653 1/20 0.56
RELA Q04206 1/20 0.56
MAPK14 Q16539 2/20 0.47
MAPK13 O15264 1/20 0.47
MAPK12 P53778 1/20 0.47
MAPK11 Q15759 1/20 0.47
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
HPGD P15428 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854348 0.90 RAB9A (0.54) RAB9ANPC1PKMALDH1A1SMN1; SMN2
SCHEMBL2852384 0.89 NPC1 (0.54) RAB9ANPC1PKMALDH1A1SMN1; SMN2
SCHEMBL2860400 0.88 RAB9A (0.53) RAB9ANPC1PKMSMN1; SMN2CYP1A2
SCHEMBL2857558 0.87 NPC1 (0.50) RAB9ANPC1PKMALDH1A1SMN1; SMN2
SCHEMBL2853093 0.87 NPC1 (0.52) RAB9ANPC1PKMALDH1A1SMN1; SMN2
SCHEMBL2855794 0.85 RAB9A (0.48) RAB9ANPC1PKMALDH1A1SMN1; SMN2
SCHEMBL2852417 0.84 MAPT (0.49) RAB9ANPC1PKMALDH1A1SMN1; SMN2
SCHEMBL2860234 0.83 HPGD (0.54) RAB9ANPC1PKMALDH1A1SMN1; SMN2
SCHEMBL2848335 0.82 ATM (0.54) RAB9ANPC1PKMSMN1; SMN2MAPT
SCHEMBL2859099 0.82 NPC1 (0.50) RAB9ANPC1PKMALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed