SCHEMBL2853093

SCHEMBL2853093

COc1ccc(-n2ncc(OC(=O)Nc3ccc(C(C)(C)C)cc3)c2C)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.52
RAB9A P51151 3/20 0.52
PKM P14618 1/20 0.52
NR1I2 O75469 2/20 0.47
NPBWR1 P48145 1/20 0.47
MCHR1 Q99705 1/20 0.47
TRPV1 Q8NER1 1/20 0.45
MAPT P10636 6/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
LPL P06858 1/20 0.44
LIPC P11150 1/20 0.44
LIPE Q05469 1/20 0.44
ALDH1A1 P00352 3/20 0.41
HTT P42858 2/20 0.41
MAPK13 O15264 1/20 0.41
MAPK12 P53778 1/20 0.41
MAPK11 Q15759 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2857953 0.88 RAB9A (0.50) NPC1RAB9APKMMAPTSMN1; SMN2
SCHEMBL2852384 0.87 NPC1 (0.54) NPC1RAB9APKMNPBWR1MCHR1
SCHEMBL2850131 0.87 RAB9A (0.61) NPC1RAB9APKMMAPTSMN1; SMN2
SCHEMBL2860400 0.86 RAB9A (0.53) NPC1RAB9APKMNPBWR1MCHR1
SCHEMBL2857558 0.79 NPC1 (0.50) NPC1RAB9APKMNPBWR1MCHR1
SCHEMBL2855794 0.77 RAB9A (0.48) NPC1RAB9APKMMAPTSMN1; SMN2
SCHEMBL2854348 0.77 RAB9A (0.54) NPC1RAB9APKMMAPTSMN1; SMN2
SCHEMBL2852417 0.77 MAPT (0.49) NPC1RAB9APKMNPBWR1MCHR1
SCHEMBL2856979 0.76 RAB9A (0.46) NPC1RAB9APKMMAPTSMN1; SMN2
SCHEMBL2848538 0.75 MAPT (0.45) NPC1RAB9ATRPV1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed