SCHEMBL2857558

SCHEMBL2857558

COc1ccc(-n2ncc(OC(=O)Nc3cccc(Cl)c3)c2C)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.50
RAB9A P51151 6/20 0.50
MEN1 O00255 5/20 0.48
KMT2A Q03164 5/20 0.48
PKM P14618 1/20 0.47
ATM Q13315 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
MAPT P10636 5/20 0.45
FADS1 O60427 1/20 0.45
NFKB1 P19838 1/20 0.45
NFKB2 Q00653 1/20 0.45
RELA Q04206 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45
LMNA P02545 1/20 0.44
NPBWR1 P48145 1/20 0.43
MCHR1 Q99705 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2853257 0.89 MAPT (0.53) NPC1RAB9AMEN1KMT2APKM
SCHEMBL2852384 0.87 NPC1 (0.54) NPC1RAB9AMEN1KMT2APKM
SCHEMBL2850131 0.87 RAB9A (0.61) NPC1RAB9AKMT2APKMSMN1; SMN2
SCHEMBL2855794 0.85 RAB9A (0.48) NPC1RAB9AMEN1KMT2APKM
SCHEMBL2860400 0.82 RAB9A (0.53) NPC1RAB9AMEN1KMT2APKM
SCHEMBL2852417 0.81 MAPT (0.49) NPC1RAB9AMEN1KMT2APKM
SCHEMBL2853093 0.79 NPC1 (0.52) NPC1RAB9AMEN1KMT2APKM
SCHEMBL3792715 0.78 SMN1; SMN2 (0.68) NPC1RAB9AMEN1KMT2AATM
SCHEMBL2854348 0.78 RAB9A (0.54) NPC1RAB9APKMSMN1; SMN2MAPT
SCHEMBL2848335 0.77 ATM (0.54) NPC1RAB9AMEN1KMT2APKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed