SCHEMBL2852384

SCHEMBL2852384

COc1ccc(-n2ncc(OC(=O)Nc3ccc(Cl)cc3)c2C)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.54
RAB9A P51151 2/20 0.54
PKM P14618 1/20 0.54
ATM Q13315 1/20 0.51
NR3C1 P04150 2/20 0.50
MAPT P10636 3/20 0.49
NPBWR1 P48145 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
MCHR1 Q99705 2/20 0.45
CNR1 P21554 3/20 0.45
CNR2 P34972 1/20 0.45
ALDH1A1 P00352 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HTT P42858 2/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2860400 0.90 RAB9A (0.53) NPC1RAB9APKMNR3C1NPBWR1
SCHEMBL2850131 0.89 RAB9A (0.61) NPC1RAB9APKMMAPTSMN1; SMN2
SCHEMBL2848335 0.87 ATM (0.54) NPC1RAB9APKMATMNR3C1
SCHEMBL2857558 0.87 NPC1 (0.50) NPC1RAB9APKMATMMAPT
SCHEMBL2853093 0.87 NPC1 (0.52) NPC1RAB9APKMATMNR3C1
SCHEMBL2858533 0.85 ATM (0.47) NPC1RAB9APKMATMNR3C1
SCHEMBL2854531 0.84 LMNA (0.52) NPC1RAB9ANR3C1MAPTNPBWR1
SCHEMBL2852417 0.83 MAPT (0.49) NPC1RAB9APKMMAPTNPBWR1
SCHEMBL2861643 0.82 CNR1 (0.50) NPC1RAB9AATMSMN1; SMN2CNR1
SCHEMBL2855794 0.79 RAB9A (0.48) NPC1RAB9APKMMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed