SCHEMBL2850834

SCHEMBL2850834

COc1ccc(Cl)c(NC(=O)Oc2cnn(-c3ccc(Cl)cc3)c2C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.45
PPARG P37231 1/20 0.41
NPBWR1 P48145 5/20 0.41
CYP3A4 P08684 4/20 0.40
CYP2C19 P33261 4/20 0.40
CYP1A2 P05177 3/20 0.40
CYP2D6 P10635 3/20 0.40
PTGS2 P35354 3/20 0.39
PTGS1 P23219 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
THPO P40225 1/20 0.39
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39
HIF1A Q16665 1/20 0.39
MAPT P10636 3/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
BRAF P15056 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2850337 0.92 MAPT (0.40) NTRK1PPARGNPBWR1CYP3A4CYP2C19
SCHEMBL2857582 0.89 MAPT (0.42) NTRK1NPBWR1NPSR1MAPTKMT2A
SCHEMBL2860522 0.87 MAPT (0.48) NTRK1CYP3A4CYP2C19CYP1A2NPSR1
SCHEMBL2858533 0.86 ATM (0.47) NPBWR1CYP3A4CYP2C19CYP1A2PTGS2
SCHEMBL2858311 0.85 RAB9A (0.47) CYP3A4CYP2C19CYP2C9TSHRMAPT
SCHEMBL2854533 0.84 MEN1 (0.46) CYP3A4CYP2C19CYP1A2NPSR1CYP2C9
SCHEMBL2852552 0.84 MEN1 (0.51) NPSR1MAPTKMT2AMEN1ALDH1A1
SCHEMBL2859712 0.83 CA1 (0.45) PTGS2PTGS1MAPTSMN1; SMN2
SCHEMBL2850809 0.82 MAPT (0.43) NPSR1TSHRMAPTKMT2AALDH1A1
SCHEMBL2859050 0.82 PTGS1 (0.46) NTRK1NPBWR1CYP3A4CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed