SCHEMBL2859050

SCHEMBL2859050

COc1ccc(OC(=O)Nc2cnn(-c3ccc(Cl)cc3)c2C(F)(F)F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.46
PTGS2 P35354 2/20 0.46
NPSR1 Q6W5P4 2/20 0.46
TSHR P16473 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
THPO P40225 1/20 0.46
BLM P54132 1/20 0.46
PMP22 Q01453 1/20 0.46
HIF1A Q16665 1/20 0.46
NPBWR1 P48145 3/20 0.45
MALT1 Q9UDY8 1/20 0.43
MAPT P10636 4/20 0.42
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
HTT P42858 4/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
KMT2A Q03164 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2859651 0.89 MAPT (0.46) NPSR1MAPTNPC1RAB9AHTT
SCHEMBL2856049 0.85 ATM (0.53) NPSR1TSHRMAPTNPC1RAB9A
SCHEMBL2858533 0.83 ATM (0.47) PTGS1PTGS2NPSR1TSHRCYP1A2
SCHEMBL2850834 0.82 NTRK1 (0.45) PTGS1PTGS2NPSR1TSHRCYP1A2
SCHEMBL2850337 0.81 MAPT (0.40) PTGS1PTGS2NPSR1TSHRCYP1A2
SCHEMBL2858063 0.80 MAPT (0.57) NPSR1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL2856664 0.80 CYP1A2 (0.55) CYP1A2CYP3A4CYP2C19MAPTNPC1
SCHEMBL2859797 0.80 MAPT (0.49) NPSR1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL2850038 0.79 MAPT (0.46) NPSR1TSHRMAPTNPC1RAB9A
SCHEMBL2854156 0.77 ROCK2 (0.46) NPSR1TSHRCYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed