SCHEMBL28513264

SCHEMBL28513264

O=C(NCCc1cccc(F)c1)c1ccc2nc(-c3ccccc3)n(Cc3ccccc3)c2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.53
GAA P10253 1/20 0.53
LMNA P02545 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
CYP11B2 P19099 1/20 0.51
BRD4 O60885 2/20 0.49
NAMPT P43490 2/20 0.48
POLB P06746 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
PDE2A O00408 2/20 0.47
PDE10A Q9Y233 1/20 0.47
MAPT P10636 2/20 0.47
ALDH1A1 P00352 2/20 0.46
PDE6D O43924 1/20 0.46
ALDH2 P05091 1/20 0.46
ALDH3A1 P30838 1/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
MMP2 P08253 1/20 0.45
MMP9 P14780 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28510581 0.83 SMN1; SMN2 (0.59) TP53CYP11B2SMN1; SMN2PDE2AMAPT
SCHEMBL28516171 0.83 THRB (0.50) TP53TDP1BRD4NAMPTSMN1; SMN2
SCHEMBL28507636 0.82 ACSS2 (0.59) TP53LMNABRD4PDE2AALDH1A1
Trifluoroacetic Acid SCHEMBL15568526 0.80 MAPT (0.58) TP53TDP1BRD4SMN1; SMN2MAPT
SCHEMBL28514126 0.80 PDE6D (0.47) TP53GAACYP11B2BRD4NAMPT
SCHEMBL28503579 0.78 ALDH1A1 (0.63) TP53LMNACYP11B2BRD4SMN1; SMN2
SCHEMBL28503584 0.78 PIK3CA (0.62) GAAPOLBPDE2AMAPTALDH1A1
Trifluoroacetic Acid SCHEMBL15569065 0.78 MAPT (0.56) TP53GAALMNAPOLBSMN1; SMN2
SCHEMBL28505411 0.75 DRD2 (0.66) TP53LMNACYP11B2BRD4SMN1; SMN2
SCHEMBL28505485 0.75 PPARG (0.58) GAALMNABRD4ALDH1A1PDE6D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107311933-B Benzimidazole derivative, preparation method and application thereof 中国人民解放军军事医学科学院毒物药物研究所 2020-12-22 CN disclosed