SCHEMBL2852350

SCHEMBL2852350

Cc1c(OC(=O)NCCc2ccccc2)cnn1-c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
HPGD P15428 1/20 0.52
TAAR1 Q96RJ0 2/20 0.50
GAA P10253 2/20 0.50
CNR1 P21554 1/20 0.48
CNR2 P34972 1/20 0.48
TP53 P04637 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
NR3C1 P04150 1/20 0.45
MAPK1 P28482 1/20 0.45
MAPT P10636 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2859872 0.92 TAAR1 (0.54) NPC1RAB9AHPGDTAAR1GAA
SCHEMBL2854887 0.92 HPGD (0.49) NPC1RAB9AHPGDNR3C1
SCHEMBL2853389 0.91 NPC1 (0.62) NPC1RAB9ATAAR1GAATP53
SCHEMBL2861261 0.88 HPGD (0.64) NPC1RAB9AHPGDGAAMAPK1
SCHEMBL2861634 0.87 RAB9A (0.44) NPC1RAB9AHPGDTAAR1TP53
SCHEMBL2857468 0.86 MAPT (0.47) NPC1RAB9AHPGDTP53L3MBTL1
SCHEMBL2856602 0.85 RIPK1 (0.46) HPGDTP53MAPK1MAPT
SCHEMBL2856862 0.84 NPC1 (0.53) NPC1RAB9ATAAR1GAAMAPT
SCHEMBL2857276 0.84 RAB9A (0.47) NPC1RAB9AHPGDTP53MAPK1
SCHEMBL2854509 0.83 KDM4E (0.50) NPC1RAB9ATAAR1GAATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed