SCHEMBL2856602

SCHEMBL2856602

Cc1c(OC(=O)NCCc2ccccc2Cl)cnn1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.46
TP53 P04637 2/20 0.45
P2RX7 Q99572 5/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HIF1A Q16665 2/20 0.44
ABCB11 O95342 1/20 0.44
HPGD P15428 1/20 0.42
MAPT P10636 1/20 0.41
USP2 O75604 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2858680 0.91 NPC1 (0.45) TP53P2RX7KMT2AABCB11MAPT
SCHEMBL2854704 0.90 P2RX7 (0.48) TP53P2RX7MEN1KMT2AHPGD
SCHEMBL2861634 0.89 RAB9A (0.44) TP53HPGDMAPTMAPK1
SCHEMBL2858097 0.89 P2RX7 (0.53) TP53P2RX7HPGDMAPT
SCHEMBL2852350 0.85 NPC1 (0.53) TP53HPGDMAPTMAPK1
SCHEMBL2859872 0.85 TAAR1 (0.54) TP53MEN1KMT2AHPGD
SCHEMBL2856697 0.85 KDM4E (0.46) RIPK1TP53P2RX7HIF1AABCB11
SCHEMBL2857276 0.83 RAB9A (0.47) TP53P2RX7HPGDMAPTMAPK1
SCHEMBL2850369 0.81 P2RX7 (0.56) TP53P2RX7MAPT
SCHEMBL2858580 0.81 HIF1A (0.43) TP53P2RX7HIF1AMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed