SCHEMBL2852799

SCHEMBL2852799

Cc1cccc(NC(=O)Oc2cnn(-c3ccc(F)cc3)c2C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
FAAH O00519 1/20 0.46
CYP3A4 P08684 1/20 0.46
MAPK1 P28482 1/20 0.46
RXFP1 Q9HBX9 1/20 0.45
NPY5R Q15761 1/20 0.43
DRD4 P21917 1/20 0.43
KDM4E B2RXH2 2/20 0.42
HPGD P15428 1/20 0.42
RAB9A P51151 2/20 0.41
NPC1 O15118 1/20 0.41
NR3C1 P04150 2/20 0.41
BRAF P15056 1/20 0.41
CCR1 P32246 1/20 0.41
LMNA P02545 2/20 0.41
MAPT P10636 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HTT P42858 1/20 0.40
TP53 P04637 1/20 0.40
P2RX7 Q99572 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2853258 0.91 NPY5R (0.45) ALDH1A1FAAHCYP3A4MAPK1NPY5R
SCHEMBL2854269 0.91 RAB9A (0.46) ALDH1A1RAB9ANPC1BRAFCCR1
SCHEMBL2856385 0.87 CCR1 (0.44) RXFP1RAB9ABRAFCCR1LMNA
SCHEMBL2861572 0.85 CA1 (0.49)
SCHEMBL2854572 0.84 RAB9A (0.44) CYP3A4KDM4ERAB9ANPC1BRAF
SCHEMBL2852361 0.84 KDM4E (0.47) ALDH1A1MAPK1NPY5RKDM4EHPGD
SCHEMBL2850550 0.83 CCR1 (0.54) KDM4ECCR1P2RX7
SCHEMBL2850032 0.82 NPC1 (0.56) ALDH1A1RXFP1NPY5RKDM4ERAB9A
SCHEMBL2861646 0.82 NPC1 (0.42) NPY5RKDM4ERAB9ANPC1BRAF
SCHEMBL2850258 0.82 MAPT (0.51) CYP3A4NPY5RKDM4EHPGDBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed