SCHEMBL2852972

SCHEMBL2852972

O=C(NC1CCCC1)c1cnn(-c2ccc([N+](=O)[O-])cc2)c1C(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SPR P35270 1/20 0.52
HSD11B1 P28845 2/20 0.51
ACHE P22303 3/20 0.51
MAPT P10636 3/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 1/20 0.47
CCR1 P32246 1/20 0.45
DDR1 Q08345 1/20 0.45
MAPK11 Q15759 1/20 0.45
MAPK14 Q16539 1/20 0.45
DDR2 Q16832 1/20 0.45
TMEM97 Q5BJF2 1/20 0.45
MAP3K20 Q9NYL2 1/20 0.45
MAP3K2 Q9Y2U5 1/20 0.45
EPHX1 P07099 1/20 0.44
POLB P06746 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2860624 0.86 SPR (0.57) SPRHSD11B1MAPTALDH1A1KDM4E
SCHEMBL2851938 0.85 SPR (0.56) SPRHSD11B1ACHEMAPTNPC1
SCHEMBL2852540 0.85 KDM4E (0.66) SPRHSD11B1MAPTNPSR1ALDH1A1
SCHEMBL2856647 0.84 MAPK11 (0.52) HSD11B1ACHEMAPTNPC1RAB9A
SCHEMBL2854367 0.82 SPR (0.56) SPRHSD11B1MAPTNPC1RAB9A
SCHEMBL2856308 0.82 SPR (0.51) SPRHSD11B1NPC1RAB9AALDH1A1
SCHEMBL2854458 0.81 ACHE (0.56) HSD11B1ACHEMAPTNPC1RAB9A
SCHEMBL10366974 0.80 HSD11B1 (0.56) SPRHSD11B1ACHEMAPTNPC1
SCHEMBL10364638 0.80 NPC1 (0.59) SPRHSD11B1MAPTNPC1RAB9A
SCHEMBL10365365 0.80 ALDH1A1 (0.69) SPRHSD11B1MAPTNPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed