SCHEMBL2853334

SCHEMBL2853334

O=C(NCc1ccc(C(F)(F)F)cc1)Oc1cnn(-c2ccc(Cl)cc2)c1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 6/20 0.47
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
MAPT P10636 2/20 0.41
P2RX7 Q99572 1/20 0.41
PTGER4 P35408 1/20 0.40
MAPK1 P28482 1/20 0.40
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
PTGES O14684 1/20 0.39
HSP90AA1 P07900 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TRPC3 Q13507 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854322 0.92 ABCB1 (0.45) CCR1MAPTP2RX7MAPK1ALDH1A1
SCHEMBL2850425 0.92 P2RX7 (0.49) CCR1MAPTP2RX7MAPK1NPSR1
SCHEMBL2853270 0.91 CCR1 (0.51) CCR1MAPTP2RX7HSP90AA1NPSR1
SCHEMBL2853388 0.91 CCR1 (0.48) CCR1CNR2MAPTP2RX7ALDH1A1
SCHEMBL2856356 0.91 ALDH1A1 (0.47) CCR1MAPTALDH1A1HPGDNPSR1
SCHEMBL2859091 0.91 CCR1 (0.46) CCR1P2RX7MAPK1
SCHEMBL2852454 0.90 KDM4E (0.48) CCR1MAPTPTGER4ALDH1A1HPGD
SCHEMBL2860715 0.90 ALDH1A1 (0.46) CCR1MAPTALDH1A1HPGD
SCHEMBL2858209 0.89 CCR1 (0.48) CCR1CNR1CNR2P2RX7MAPK1
SCHEMBL2848661 0.89 ABCB1 (0.48) CCR1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed