SCHEMBL2856356

SCHEMBL2856356

O=C(NCc1ccc(Cl)cc1)Oc1cnn(-c2ccccc2)c1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.46
MAPT P10636 2/20 0.46
POLB P06746 1/20 0.46
TP53 P04637 3/20 0.45
GAA P10253 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
MAPK11 Q15759 2/20 0.45
MAPK14 Q16539 2/20 0.45
DDR1 Q08345 1/20 0.45
DDR2 Q16832 1/20 0.45
TMEM97 Q5BJF2 1/20 0.45
MAP3K20 Q9NYL2 1/20 0.45
MAP3K2 Q9Y2U5 1/20 0.45
CCR1 P32246 4/20 0.43
NR3C1 P04150 1/20 0.43
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2853388 0.96 CCR1 (0.48) ALDH1A1KDM4ESMN1; SMN2MAPTPOLB
SCHEMBL2861243 0.92 KDM4E (0.52) ALDH1A1KDM4ESMN1; SMN2MAPTPOLB
SCHEMBL2853334 0.91 CCR1 (0.47) ALDH1A1MAPTCCR1NPSR1HPGD
SCHEMBL2850425 0.91 P2RX7 (0.49) MAPTPOLBTP53CCR1NPSR1
SCHEMBL2854847 0.91 ALDH1A1 (0.48) ALDH1A1KDM4ESMN1; SMN2MAPTPOLB
SCHEMBL2852454 0.91 KDM4E (0.48) ALDH1A1KDM4ESMN1; SMN2MAPTPOLB
SCHEMBL2859861 0.90 TAAR1 (0.51) ALDH1A1KDM4ESMN1; SMN2MAPTPOLB
SCHEMBL2857598 0.90 KMT2A (0.48) ALDH1A1KDM4ESMN1; SMN2MAPTPOLB
SCHEMBL2859307 0.89 TSHR (0.46) ALDH1A1KDM4ESMN1; SMN2MAPTPOLB
SCHEMBL2854322 0.89 ABCB1 (0.45) ALDH1A1KDM4ESMN1; SMN2MAPTMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed