SCHEMBL28534028

SCHEMBL28534028

CCOC(=O)CCCN(OC(=O)C1CC1)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 1/20 0.39
TSHR P16473 1/20 0.39
KMT2A Q03164 1/20 0.39
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
CYP1A2 P05177 1/20 0.36
HDAC6 Q9UBN7 2/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
MAPT P10636 2/20 0.35
SMYD3 Q9H7B4 1/20 0.34
USP2 O75604 1/20 0.34
ALOX15 P16050 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
HSD11B1 P28845 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29239679 0.80 L3MBTL1 (0.36) ALDH1A1MEN1TSHRKMT2ANFKB1
SCHEMBL27833367 0.78 NFKB1 (0.37) ALDH1A1MEN1TSHRKMT2ANFKB1
SCHEMBL29239760 0.77 HRH3 (0.34) ALDH1A1MEN1TSHRKMT2ANFKB1
SCHEMBL19784442 0.76 HDAC6 (0.42) ALDH1A1TSHRKMT2ACYP1A2HDAC6
SCHEMBL29285429 0.75 CA14 (0.47) ALDH1A1TSHRNFKB1NFKB2RELA
SCHEMBL11031396 0.75 ALDH1A1 (0.47) ALDH1A1MEN1TSHRKMT2AMAPT
SCHEMBL14822004 0.74 CYP1A2 (0.44) ALDH1A1TSHRNFKB1NFKB2RELA
SCHEMBL1771789 0.73 BTK (0.37) ALDH1A1MEN1TSHRKMT2ANFKB1
SCHEMBL28612600 0.72 KMT2A (0.38) ALDH1A1MEN1TSHRKMT2ANFKB1
SCHEMBL1296762 0.71 ALDH1A1 (0.55) ALDH1A1MEN1TSHRKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113767103-A Novel spirocyclic K-Ras G12C inhibitor 微境生物医药科技(上海)有限公司 2021-12-07 CN disclosed
CN-112390797-A Novel spirocyclic K-Ras G12C inhibitor 微境生物医药科技(上海)有限公司 2021-02-23 CN disclosed