SCHEMBL2854430

SCHEMBL2854430

O=C(NCC1CCCCC1)c1cnn(-c2ccc(Cl)nn2)c1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK11 Q15759 2/20 0.47
MAPK14 Q16539 2/20 0.47
DDR1 Q08345 1/20 0.47
DDR2 Q16832 1/20 0.47
TMEM97 Q5BJF2 1/20 0.47
MAP3K20 Q9NYL2 1/20 0.47
MAP3K2 Q9Y2U5 1/20 0.47
P2RX7 Q99572 1/20 0.46
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
CNR2 P34972 5/20 0.44
HDAC6 Q9UBN7 5/20 0.44
CYP3A4 P08684 3/20 0.43
CYP2C9 P11712 3/20 0.43
CYP2C19 P33261 3/20 0.43
CYP1A2 P05177 2/20 0.42
MLYCD O95822 1/20 0.42
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HDAC3 O15379 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2850365 0.84 SPR (0.53) MAPK11MAPK14DDR1DDR2TMEM97
SCHEMBL2854446 0.83 MAPK11 (0.55) MAPK11MAPK14DDR1DDR2TMEM97
SCHEMBL2852950 0.81 MAPK14 (0.67) MAPK11MAPK14DDR1DDR2TMEM97
SCHEMBL2853007 0.80 MAPK11 (0.58) MAPK11MAPK14DDR1DDR2TMEM97
SCHEMBL2856270 0.80 MAPK14 (0.56) MAPK11MAPK14DDR1DDR2TMEM97
SCHEMBL2850254 0.80 CNR2 (0.52) MAPK11MAPK14DDR1DDR2TMEM97
SCHEMBL2852810 0.77 KDM4E (0.48) MAPK11MAPK14DDR1DDR2TMEM97
SCHEMBL2856252 0.77 P2RX1 (0.49) MLYCDTRPC3
SCHEMBL2855644 0.77 ALDH1A1 (0.44) KDM4EALDH1A1TRPC3KMT2AMAPT
SCHEMBL2848180 0.77 CCR1 (0.51) MAPK11MAPK14DDR1DDR2TMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed