SCHEMBL2854450

SCHEMBL2854450

Cc1c(OC(=O)NC2CCN(c3ccc(OC(F)(F)F)cc3)C2)cnn1-c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 7/20 0.46
CASR P41180 2/20 0.43
SMPD3 Q9NY59 1/20 0.41
CCNC P24863 3/20 0.41
CDK8 P49336 3/20 0.41
NOTUM Q6P988 1/20 0.41
CHRM2 P08172 2/20 0.41
CHRM1 P11229 2/20 0.41
ABL1 P00519 1/20 0.40
BCR P11274 1/20 0.40
EPHX2 P34913 1/20 0.40
MAPT P10636 2/20 0.39
NPC1 O15118 1/20 0.39
NFKB1 P19838 1/20 0.39
RAB9A P51151 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM3 P20309 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2857649 0.92 NOTUM (0.51) CHRM4CASRNOTUMCHRM2CHRM1
SCHEMBL2854779 0.84 SMO (0.49) CASRNOTUM
SCHEMBL2859595 0.78 CHRM4 (0.53) CHRM4CHRM2CHRM1CHRM5CHRM3
SCHEMBL22815701 0.75 CHRM4 (0.49) CHRM4CASRSMPD3CCNCCDK8
SCHEMBL14989237 0.74 MAPK13 (0.44) MAPTNPC1NFKB1RAB9ANFKB2
SCHEMBL2854465 0.72 RAB9A (0.47) MAPTNPC1NFKB1RAB9ANFKB2
SCHEMBL31288311 0.71 CHRM4 (0.58) CHRM4EPHX2MAPTSMN1; SMN2
SCHEMBL5138185 0.71 FAAH (0.41) MAPTRAB9ASMN1; SMN2
SCHEMBL2856979 0.70 RAB9A (0.46) MAPTNPC1NFKB1RAB9ANFKB2
SCHEMBL23484542 0.70 MAP4K4 (0.49) CHRM4EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed