SCHEMBL2859595

SCHEMBL2859595

O=C(NC1CCN(Cc2ccccc2)C1)Oc1cnn(-c2ccc(OC(F)(F)F)cc2)c1C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 12/20 0.53
BCHE P06276 2/20 0.52
ACHE P22303 2/20 0.52
BACE1 P56817 2/20 0.52
CCR2 P41597 1/20 0.49
CHRM2 P08172 2/20 0.47
CHRM1 P11229 2/20 0.47
CHRM5 P08912 1/20 0.47
CHRM3 P20309 1/20 0.47
DRD4 P21917 3/20 0.47
HTR2A P28223 2/20 0.47
DRD2 P14416 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854763 0.91 DRD4 (0.50) BCHEACHEBACE1CCR2DRD4
SCHEMBL2857724 0.86 SIGMAR1 (0.53) CHRM4
SCHEMBL2863246 0.85 DRD4 (0.49) CCR2DRD4DRD2
SCHEMBL2858617 0.85 CHRM4 (0.58) CHRM4BCHEACHEBACE1CHRM2
SCHEMBL2857980 0.84 DRD4 (0.47) CHRM4CCR2DRD4DRD2
SCHEMBL2856452 0.83 DRD4 (0.47) CCR2DRD4DRD2
SCHEMBL2854450 0.78 CHRM4 (0.46) CHRM4CHRM2CHRM1CHRM5CHRM3
SCHEMBL2854556 0.76 DRD4 (0.47) BACE1DRD4DRD2
SCHEMBL2852970 0.75 DRD2 (0.51) CCR2DRD4DRD2
SCHEMBL25153723 0.74 EPHX2 (0.73) CHRM4BCHEACHEBACE1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed