SCHEMBL2854556

SCHEMBL2854556

CCCc1c(OC(=O)NC2CCN(Cc3ccccc3)C2)cnn1-c1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 8/20 0.47
DRD2 P14416 5/20 0.47
MCHR1 Q99705 1/20 0.46
BACE1 P56817 1/20 0.44
MME P08473 1/20 0.44
SIGMAR1 Q99720 1/20 0.43
DPP7 Q9UHL4 1/20 0.43
MC4R P32245 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15889273 0.79 POLB (0.58) DRD4SIGMAR1
SCHEMBL2854763 0.78 DRD4 (0.50) DRD4DRD2BACE1SIGMAR1
SCHEMBL2859595 0.76 CHRM4 (0.53) DRD4DRD2BACE1
SCHEMBL2863246 0.76 DRD4 (0.49) DRD4DRD2MCHR1SIGMAR1
SCHEMBL2854713 0.75 NTRK1 (0.49)
SCHEMBL10155707 0.75 MCHR1 (0.61) DRD4DRD2MCHR1SIGMAR1
SCHEMBL2856997 0.74 ALDH1A1 (0.57)
SCHEMBL2857980 0.74 DRD4 (0.47) DRD4DRD2MCHR1SIGMAR1
SCHEMBL2850487 0.74 HTT (0.48)
SCHEMBL2856452 0.74 DRD4 (0.47) DRD4DRD2MCHR1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed