SCHEMBL2850487

SCHEMBL2850487

CCCc1c(OC(=O)NC2CCCc3ccccc32)cnn1-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.48
ALDH1A1 P00352 5/20 0.47
NTRK1 P04629 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
CNR1 P21554 1/20 0.45
CNR2 P34972 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
TAOK1 Q7L7X3 1/20 0.44
TAOK3 Q9H2K8 1/20 0.44
MAPK1 P28482 1/20 0.44
TAS1R3 Q7RTX0 1/20 0.43
TAS1R1 Q7RTX1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854713 0.94 NTRK1 (0.49) HTTALDH1A1NTRK1MEN1KMT2A
SCHEMBL2850723 0.93 TAOK3 (0.47) HTTALDH1A1SMN1; SMN2L3MBTL1CNR2
SCHEMBL2860851 0.88 CNR1 (0.46) HTTALDH1A1NTRK1SMN1; SMN2CNR1
SCHEMBL2854219 0.82 ALDH1A1 (0.47) HTTALDH1A1NTRK1SMN1; SMN2MEN1
SCHEMBL2857348 0.78 SPR (0.54) ALDH1A1NTRK1MAPK1TAS1R3TAS1R1
SCHEMBL2852199 0.76 KMT2A (0.47) HTTALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL2860401 0.76 MAPK13 (0.47) HTTALDH1A1NTRK1SMN1; SMN2MAPK1
SCHEMBL3395550 0.76 SPR (0.55) ALDH1A1CNR2TAS1R3TAS1R1
SCHEMBL2857660 0.76 LMNA (0.48) HTTALDH1A1SMN1; SMN2CNR1MEN1
SCHEMBL3391804 0.76 SPR (0.55) ALDH1A1CNR2TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed