SCHEMBL2854713

SCHEMBL2854713

CCCc1c(OC(=O)NC2CCc3ccccc32)cnn1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 3/20 0.49
MAPK13 O15264 1/20 0.45
MAPK12 P53778 1/20 0.45
MAPK11 Q15759 1/20 0.45
MAPK14 Q16539 1/20 0.45
ALDH1A1 P00352 6/20 0.42
MAPK1 P28482 2/20 0.42
MAPT P10636 3/20 0.41
EPHX2 P34913 2/20 0.41
PDE2A O00408 1/20 0.41
HTT P42858 2/20 0.41
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
SPR P35270 1/20 0.40
RAB9A P51151 1/20 0.40
GAA P10253 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2850487 0.94 HTT (0.48) NTRK1ALDH1A1MAPK1HTTMEN1
SCHEMBL2860851 0.93 CNR1 (0.46) NTRK1MAPK13MAPK12MAPK11MAPK14
SCHEMBL2850723 0.88 TAOK3 (0.47) ALDH1A1HTTMEN1KMT2A
SCHEMBL2857348 0.83 SPR (0.54) NTRK1MAPK14ALDH1A1MAPK1MAPT
SCHEMBL2860401 0.82 MAPK13 (0.47) NTRK1MAPK13MAPK12MAPK11MAPK14
SCHEMBL2852200 0.77 SPR (0.51) MAPK14ALDH1A1MAPK1MAPTPDE2A
SCHEMBL2856997 0.76 ALDH1A1 (0.57) MAPK14ALDH1A1MAPK1MAPTRAB9A
SCHEMBL2854219 0.76 ALDH1A1 (0.47) NTRK1ALDH1A1MAPK1MAPTHTT
SCHEMBL5325459 0.76 ALDH1A1 (0.53) MAPK14ALDH1A1MAPK1MAPTRAB9A
SCHEMBL2854556 0.75 DRD4 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed