SCHEMBL2854804

SCHEMBL2854804

O=C(NCc1ccccc1)Oc1cnn(-c2ccc(F)cc2)c1C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.48
CCR1 P32246 6/20 0.47
P2RX7 Q99572 1/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
SMO Q99835 2/20 0.45
TP53 P04637 2/20 0.45
MAPT P10636 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
POLB P06746 1/20 0.44
RAB9A P51151 1/20 0.44
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854847 0.96 ALDH1A1 (0.48) MAPK1CCR1P2RX7KDM4EALDH1A1
SCHEMBL2861243 0.93 KDM4E (0.52) CCR1KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL2860715 0.92 ALDH1A1 (0.46) CCR1KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL2853388 0.91 CCR1 (0.48) CCR1P2RX7KDM4EALDH1A1TP53
SCHEMBL2859091 0.91 CCR1 (0.46) MAPK1CCR1P2RX7SMORAB9A
SCHEMBL2855710 0.90 LMNA (0.46) MAPK1CCR1P2RX7SMOMAPT
SCHEMBL2854346 0.90 MAPT (0.52) MAPK1CCR1P2RX7KDM4EALDH1A1
SCHEMBL2850425 0.90 P2RX7 (0.49) MAPK1CCR1P2RX7SMOTP53
SCHEMBL2853351 0.89 CCR1 (0.62) CCR1P2RX7KDM4E
SCHEMBL2852520 0.89 TP53 (0.47) MAPK1KDM4EALDH1A1TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed