SCHEMBL2854814

SCHEMBL2854814

Cc1cccc(CNC(=O)Oc2cnn(-c3ccccc3)c2C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.47
CCR1 P32246 5/20 0.46
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
DDT P30046 1/20 0.44
HPGD P15428 1/20 0.44
POLB P06746 1/20 0.44
MAPT P10636 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KEAP1 Q14145 1/20 0.44
NFE2L2 Q16236 1/20 0.44
KMT2A Q03164 2/20 0.41
METAP2 P50579 1/20 0.41
LMNA P02545 1/20 0.41
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2850550 0.92 CCR1 (0.54) CCR1KDM4EDDT
SCHEMBL2854543 0.92 CCR1 (0.54) TP53CCR1DDTMAPTKMT2A
SCHEMBL2861243 0.90 KDM4E (0.52) CCR1KDM4EALDH1A1HPGDPOLB
SCHEMBL2860247 0.89 CCR1 (0.59) CCR1KDM4EALDH1A1POLBMAPT
SCHEMBL2856304 0.89 KEAP1 (0.53) CCR1KDM4EALDH1A1HPGDPOLB
SCHEMBL2857598 0.89 KMT2A (0.48) KDM4EALDH1A1HPGDPOLBMAPT
SCHEMBL2857073 0.85 CCR1 (0.48) CCR1KDM4EALDH1A1POLBMAPT
SCHEMBL2859307 0.84 TSHR (0.46) CCR1KDM4EALDH1A1POLBMAPT
SCHEMBL2854462 0.84 KEAP1 (0.48) CCR1KDM4EALDH1A1MAPTKEAP1
SCHEMBL2854847 0.84 ALDH1A1 (0.48) TP53CCR1KDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed