SCHEMBL28560281

SCHEMBL28560281

CNc1ccc([N+](=O)[O-])c(Cl)c1Cl

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.57
HCAR3 P49019 1/20 0.47
CRHBP P24387 1/20 0.47
CRHR2 Q13324 1/20 0.47
HTT P42858 1/20 0.45
MAPT P10636 5/20 0.44
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTR2A P28223 2/20 0.41
HTR2C P28335 2/20 0.41
HTR2B P41595 2/20 0.41
TSHR P16473 2/20 0.41
MAPK1 P28482 1/20 0.41
POLB P06746 1/20 0.41
CDC25B P30305 1/20 0.40
GPR35 Q9HC97 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21461475 0.84 TDP1 (0.47) TDP1HCAR3CRHBPCRHR2HTT
SCHEMBL28391943 0.81 TDP1 (0.81) TDP1ALDH1A1CYP1A2CYP2C9HPGD
SCHEMBL28553684 0.80 FABP3 (0.52) TDP1HCAR3CRHBPCRHR2HTT
SCHEMBL1982270 0.76 L3MBTL1 (0.61) TDP1HCAR3HTTMAPTALDH1A1
SCHEMBL487351 0.76 MAPK1 (0.58) TDP1HCAR3MAPTKMT2AALDH1A1
SCHEMBL8407132 0.75 ALDH1A1 (0.49) TDP1HCAR3HTTMAPTKMT2A
SCHEMBL1557360 0.74 HCAR3 (0.49) TDP1HCAR3HTTMAPTKMT2A
SCHEMBL5635692 0.74 TDP1 (0.63) TDP1CRHBPCRHR2MAPTKMT2A
SCHEMBL278488 0.73 TDP1 (1.00) TDP1ALDH1A1HPGDHTR2AHTR2C
SCHEMBL27707234 0.72 VCAM1 (0.42) TDP1HCAR3HTTMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112745237-B 2-arylamine compound and preparation method and application thereof 中国科学院上海药物研究所 2023-06-20 CN disclosed
CN-112745237-A 2-arylamine compound and preparation method and application thereof 中国科学院上海药物研究所 2021-05-04 CN disclosed