SCHEMBL2856049

SCHEMBL2856049

COc1ccccc1OC(=O)Nc1cnn(-c2ccc(Cl)cc2)c1C(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.53
MAPT P10636 8/20 0.42
ALDH1A1 P00352 5/20 0.42
KDM4E B2RXH2 3/20 0.42
LMNA P02545 2/20 0.42
HTT P42858 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
SCN5A Q14524 1/20 0.42
SCN9A Q15858 1/20 0.42
NPSR1 Q6W5P4 3/20 0.41
HPGD P15428 1/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
POLB P06746 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
GPR6 P46095 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
MET P08581 1/20 0.40
MST1R Q04912 1/20 0.40
ACHE P22303 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2860020 0.86 KDM4E (0.51) MAPTALDH1A1KDM4ELMNAHTT
SCHEMBL2859050 0.85 PTGS1 (0.46) MAPTALDH1A1KDM4ELMNAHTT
SCHEMBL2859651 0.85 MAPT (0.46) MAPTALDH1A1KDM4ELMNAHTT
SCHEMBL2859508 0.82 CYP1A2 (0.46) MAPTALDH1A1KDM4EHTTTDP1
SCHEMBL2856759 0.81 ACLY (0.44) ATMMAPTALDH1A1KDM4ELMNA
SCHEMBL2852552 0.81 MEN1 (0.51) MAPTALDH1A1KDM4ENPSR1SMN1; SMN2
SCHEMBL2855775 0.81 P2RY1 (0.44) ATMMAPTALDH1A1KDM4ELMNA
SCHEMBL2848541 0.80 RAB9A (0.43) MAPTALDH1A1KDM4ELMNANPSR1
SCHEMBL2854596 0.80 TP53 (0.46) MAPTALDH1A1KDM4ELMNAHTT
SCHEMBL2860986 0.80 MAPT (0.45) MAPTALDH1A1KDM4ELMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed