SCHEMBL2857017

SCHEMBL2857017

O=C(OC(=O)C(F)(F)F)c1cnn(Cc2nc(-c3cc(OCc4ccccn4)cc(C(F)(F)F)c3)cs2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PPARD Q03181 2/20 0.36
ALOX5AP P20292 3/20 0.34
MAPK14 Q16539 5/20 0.33
SMO Q99835 4/20 0.33
RHOA P61586 1/20 0.33
LDHA P00338 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
HTR2B P41595 2/20 0.32
LMNA P02545 1/20 0.32
PKM P14618 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP2C8 P10632 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2B6 P20813 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12876610 0.90 PPARD (0.39) ALDH1A1L3MBTL1PPARDALOX5APMAPK14
Trifluoroacetic Acid SCHEMBL2857015 0.90 PPARD (0.38) ALDH1A1L3MBTL1PPARDALOX5APMAPK14
SCHEMBL2858915 0.83 MAPK14 (0.35) ALOX5APMAPK14SMORHOAPPARA
SCHEMBL2860292 0.81 ALDH1A1 (0.42) ALDH1A1L3MBTL1PPARDKMT2A
SCHEMBL1198663 0.78 MMP13 (0.44) ALDH1A1L3MBTL1PPARDKMT2ASMN1; SMN2
SCHEMBL1198589 0.78 MMP13 (0.40) ALDH1A1L3MBTL1PPARDLDHAKMT2A
Trifluoroacetic Acid SCHEMBL2863073 0.77 GPR132 (0.39) ALDH1A1PPARDLDHAKMT2APPARA
SCHEMBL2861490 0.76 ALKBH1 (0.44) ALDH1A1L3MBTL1PPARDKMT2A
SCHEMBL2868652 0.76 ALKBH1 (0.45) ALDH1A1L3MBTL1PPARDKMT2A
SCHEMBL1198715 0.76 ALDH1A1 (0.42) ALDH1A1L3MBTL1PPARDKMT2APPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2264017-A1 HETEROCYCLIC DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2010-12-22 EP disclosed