SCHEMBL2853809

SCHEMBL2853809

COc1ccc(CNC(=O)Oc2cnn(-c3ccc(F)cc3)c2C(F)(F)F)c(OC)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.49
MAPT P10636 3/20 0.46
EPHX2 P34913 1/20 0.46
KLKB1 P03952 1/20 0.43
DGAT2 Q96PD7 1/20 0.43
ALDH1A1 P00352 2/20 0.43
TSHR P16473 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
PDE4B Q07343 1/20 0.42
PPARG P37231 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
TP53 P04637 1/20 0.40
GAA P10253 1/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
ROCK2 O75116 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2853175 0.92 KLKB1 (0.43) P2RX7MAPTKLKB1DGAT2ALDH1A1
SCHEMBL2852117 0.89 P2RX7 (0.48) P2RX7MAPTALDH1A1TP53GAA
SCHEMBL2860466 0.87 RCE1 (0.47) P2RX7MAPTALDH1A1TP53GAA
SCHEMBL2850896 0.86 DGAT2 (0.57) P2RX7MAPTEPHX2KLKB1DGAT2
SCHEMBL2856797 0.86 P2RX7 (0.45) P2RX7ALDH1A1
SCHEMBL2857544 0.85 TSHR (0.45) MAPTEPHX2KLKB1DGAT2ALDH1A1
SCHEMBL2853277 0.85 CCR1 (0.50) P2RX7KLKB1DGAT2TP53PKM
SCHEMBL2856615 0.84 P2RX7 (0.48) P2RX7MAPTALDH1A1NPSR1TP53
SCHEMBL2855708 0.84 P2RX7 (0.44) P2RX7MAPTDGAT2ALDH1A1NPSR1
SCHEMBL2859103 0.83 EPHX2 (0.45) MAPTEPHX2KLKB1DGAT2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed